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Found 2 Enz. Inhib. hit(s) with Target = 'Apelin receptor' and Ligand = 'BDBM50554004'
TargetApelin receptor(Rattus norvegicus)
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554004(CHEMBL4760648)
Affinity DataIC50:  6.30nMAssay Description:Displacement of [125I]-pyr-1-apelin-13 from EGFP-tagged wild-type rat apelin receptor expressed in CHO cell membranes by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50554004(CHEMBL4760648)
Affinity DataEC50:  7.80nMAssay Description:Activation of APJ receptor (unknown origin) expressed in Chem-5 cells assessed as stimulation of Ca2+ mobilization by Calcium 6-GF dye based fluoresc...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed