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Found 2 Enz. Inhib. hit(s) with Target = 'Apelin receptor' and Ligand = 'BDBM50556826'
TargetApelin receptor(Homo sapiens (Human))
Huazhong University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556826(CHEMBL4745863)
Affinity DataKi:  0.220nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Rattus norvegicus)
Huazhong University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556826(CHEMBL4745863)
Affinity DataEC50:  6.90nMAssay Description:Agonist activity at APJ receptor in rat NRK-52E cells assessed as effect on cAMP accumulation incubated for 1 hr by cAMP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed