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Found 9 Enz. Inhib. hit(s) with Target = 'Appetite-regulating hormone' and Ligand = 'BDBM50593269'
TargetAppetite-regulating hormone(Homo sapiens (Human))
Tongji University

Curated by ChEMBL
LigandPNGBDBM50593269(CHEMBL5177247)
Affinity DataIC50:  0.933nMAssay Description:Displacement of C-terminal Cys-tagged SmBiT tracer from C-terminal Cys-tagged human Ghrelin expressed in HEK293T cells by microplate reader based Nan...More data for this Ligand-Target Pair
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TargetAppetite-regulating hormone(Homo sapiens (Human))
Tongji University

Curated by ChEMBL
LigandPNGBDBM50593269(CHEMBL5177247)
Affinity DataIC50:  1.40nMAssay Description:Displacement of C-terminal Cys-tagged human LEAP2-SmBiT tracer from C-terminal Cys-tagged human Ghrelin expressed in HEK293T cells by microplate read...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetAppetite-regulating hormone(Homo sapiens (Human))
Tongji University

Curated by ChEMBL
LigandPNGBDBM50593269(CHEMBL5177247)
Affinity DataIC50:  1.5nMAssay Description:Displacement of C-terminal Cys-tagged human LEAP2-SmBiT tracer from C-terminal Cys-tagged human Ghrelin expressed in HEK293T cells by microplate read...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAppetite-regulating hormone(Bos taurus)
Tongji University

Curated by ChEMBL
LigandPNGBDBM50593269(CHEMBL5177247)
Affinity DataIC50:  9.10nMAssay Description:Binding affinity to Ghrelin in fetal bovine serum expressed in HEK293T cells using NanoLuc as substrate measured after 1 hr by bioluminescence based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAppetite-regulating hormone(Bos taurus)
Tongji University

Curated by ChEMBL
LigandPNGBDBM50593269(CHEMBL5177247)
Affinity DataIC50:  9.10nMAssay Description:Binding affinity to Ghrelin in fetal bovine serum expressed in HEK293T cells using NanoLuc as substrate measured after 1 hr by bioluminescence based ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAppetite-regulating hormone(Homo sapiens (Human))
Tongji University

Curated by ChEMBL
LigandPNGBDBM50593269(CHEMBL5177247)
Affinity DataIC50:  10nMAssay Description:Binding affinity to Ghrelin in human serum expressed in HEK293T cells using NanoLuc as substrate measured after 1 hr by bioluminescence based micropl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAppetite-regulating hormone(Homo sapiens (Human))
Tongji University

Curated by ChEMBL
LigandPNGBDBM50593269(CHEMBL5177247)
Affinity DataIC50:  11nMAssay Description:Binding affinity to Ghrelin in human serum expressed in HEK293T cells using NanoLuc as substrate measured after 1 hr by bioluminescence based micropl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAppetite-regulating hormone(Homo sapiens (Human))
Tongji University

Curated by ChEMBL
LigandPNGBDBM50593269(CHEMBL5177247)
Affinity DataEC50:  1nMAssay Description:Displacement of C-terminal Cys-tagged NanoLuc luciferase from C-terminal Cys-tagged human Ghrelin expressed in HEK293T cells by microplate reader bas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetAppetite-regulating hormone(Homo sapiens (Human))
Tongji University

Curated by ChEMBL
LigandPNGBDBM50593269(CHEMBL5177247)
Affinity DataEC50:  1nMAssay Description:Displacement of C-terminal Cys-tagged NanoLuc luciferase from C-terminal Cys-tagged human Ghrelin expressed in HEK293T cells by microplate reader bas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed