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Found 5 Enz. Inhib. hit(s) with Target = 'Arginase-1' and Ligand = 'BDBM50561034'
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561034(CHEMBL4244287)
Affinity DataIC50:  270nMAssay Description:Binding affinity to human ARG1 assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetArginase-1(Rattus norvegicus)
Oncoarendi Therapeutics

Curated by ChEMBL
LigandPNGBDBM50561034(CHEMBL4244287)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of rat Arg1 at pH 7.4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArginase-1(Rattus norvegicus)
Oncoarendi Therapeutics

Curated by ChEMBL
LigandPNGBDBM50561034(CHEMBL4244287)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of rat liver arginase using L-arginine as substrate incubated for 10 mins followed by substrate addition by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetArginase-1(Rattus norvegicus)
Oncoarendi Therapeutics

Curated by ChEMBL
LigandPNGBDBM50561034(CHEMBL4244287)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of rat ARG1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561034(CHEMBL4244287)
Affinity DataKd:  270nMAssay Description:Binding affinity to human Arg1 at pH 8.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed