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Found 2 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM50254015'
TargetAromatase(Homo sapiens (Human))
Universidade De Coimbra

Curated by ChEMBL
LigandPNGBDBM50254015(1-(2-(3,4-dichlorophenylthio)-2-(4-methoxyphenyl)e...)
Affinity DataKi:  6.5nMAssay Description:Inhibition of human aromatase-mediated conversion of [1beta3H]androstenedione to estrone by Lineweaver-Burk plot in presence of NADPHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Universidade De Coimbra

Curated by ChEMBL
LigandPNGBDBM50254015(1-(2-(3,4-dichlorophenylthio)-2-(4-methoxyphenyl)e...)
Affinity DataIC50:  25nMAssay Description:Inhibition of human aromatase-mediated conversion of [1beta3H]androstenedione to estrone by liquid scintillation counting in presence of NADPHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed