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Found 2 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM8581'
TargetAromatase(Homo sapiens (Human))
University Of Calcutta

Curated by ChEMBL
LigandPNGBDBM8581((3-Pyridylmethylene)indane 1a | 3-[(1E)-2,3-dihydr...)
Affinity DataIC50:  2.04E+3nMAssay Description:Inhibition of aromataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Calcutta

Curated by ChEMBL
LigandPNGBDBM8581((3-Pyridylmethylene)indane 1a | 3-[(1E)-2,3-dihydr...)
Affinity DataIC50:  2.04E+3nMpH: 7.4 T: 2°CAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta-3H] Androstenedione during aromatization. After incubation, the re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed