Affinity DataKi: 0.440nMAssay Description:Inhibition of human bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Displacement of [3H]des-Arg10 Leu9 kallidin from human bradykinin B1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.440nMAssay Description:Binding affinity to human BK1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to rhesus monkey bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Binding affinity to rabbit bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+3nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.65E+3nMAssay Description:Binding affinity to rat bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.52nMAssay Description:Activity at human bradykinin B1 receptor assessed as inhibition of Des-arg kallidin-induced increase of cytosolic calcium in CHO cells by FLIPRMore data for this Ligand-Target Pair