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Found 2 Enz. Inhib. hit(s) with Target = 'B1 bradykinin receptor' and Ligand = 'BDBM50264296'
TargetB1 bradykinin receptor(Macaca fascicularis)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264296(1-benzyl-N-(2-oxo-2-(4-(pyridin-4-yl)piperazin-1-y...)
Affinity DataIC50:  310nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264296(1-benzyl-N-(2-oxo-2-(4-(pyridin-4-yl)piperazin-1-y...)
Affinity DataIC50:  417nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed