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Found 2 Enz. Inhib. hit(s) with Target = 'B1 bradykinin receptor' and Ligand = 'BDBM50264298'
TargetB1 bradykinin receptor(Macaca fascicularis)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264298(CHEMBL490201 | N-(2-((4-(4,5-dihydro-1H-imidazol-2...)
Affinity DataIC50:  5nMAssay Description:Antagonist activity at Cynomolgus monkey bradykinin B1 receptor expressed in CHO cells assessed as calcium transient by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(RAT)
Neurogen

Curated by ChEMBL
LigandPNGBDBM50264298(CHEMBL490201 | N-(2-((4-(4,5-dihydro-1H-imidazol-2...)
Affinity DataIC50:  155nMAssay Description:Antagonist activity at rat bradykinin B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed