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Found 2 Enz. Inhib. hit(s) with Target = 'Beta-1 adrenergic receptor' and Ligand = 'BDBM50001884'
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Centro De InvestigacióN Grupo Ferrer

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataKi:  2.60E+4nMAssay Description:Binding affinity measured at the Beta-1 adrenergic receptor by the inhibition of [3H]-DHA binding to rat cortex using unlabeled isoprenalin for nonsp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Rattus norvegicus (Rat))
Centro De InvestigacióN Grupo Ferrer

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity against beta-1 adrenergic receptor in rat brain using [3H]-DHAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed