Found 8 Enz. Inhib. hit(s) with Target = 'Beta-2 adrenergic receptor' and Ligand = 'BDBM50167064' TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 97nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 97nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Agonist activity at human beta2 receptor expressed in HEK293 cells cotransfected with Gqs5 protein assessed as [3H]IP3 accumulation after 120 mins by...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataEC50: 269nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataEC50: 100nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataEC50: 63nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring Rluc2-117-GalphaS/GFP10-Ggamma/Gbeta1 assessed as...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataEC50: 158nMAssay Description:Agonist activity at beta2-adrenergic receptor (unknown origin) expressed in HEK293T cells harboring GFP/Rluc2-tagged beta-arrestin2 assessed as incre...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataEC50: 210nMAssay Description:Agonist activity at PK-tagged beta2 receptor (unknown origin) transfected in HEK293 cells after 90 mins by beta-arrestin assayMore data for this Ligand-Target Pair
