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Found 3 Enz. Inhib. hit(s) with Target = 'Beta-glucuronidase' and Ligand = 'BDBM178133'
TargetBeta-glucuronidase(Bos taurus (Bovine))
Universiti Teknologi Mara (Uitm), Puncak Alam Campus

LigandPNGBDBM178133(3-(6-Chloro-1H-imidazo[4,5-b]pyridin-2-yl)benzene-...)
Affinity DataIC50:  2.93E+4nMAssay Description:The protocol followed in this study was earlier reported [33,34]. β-Glucuronidase activity was evaluated by measuring the absorbance at 405 nm o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucuronidase(Homo sapiens (Human))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM178133(3-(6-Chloro-1H-imidazo[4,5-b]pyridin-2-yl)benzene-...)
Affinity DataIC50:  2.93E+4nMAssay Description:Inhibition of beta-glucuronidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucuronidase(Homo sapiens (Human))
University Of Kwazulu-Natal

Curated by ChEMBL
LigandPNGBDBM178133(3-(6-Chloro-1H-imidazo[4,5-b]pyridin-2-yl)benzene-...)
Affinity DataIC50:  2.93E+4nMAssay Description:Inhibition of beta-glucuronidase (unknown origin) using p-nitrophenyl-beta-D-glucuronide as substrate pre-incubated for 30 mins followed by substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed