Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with Target = 'Beta-lactamase' and Ligand = 'BDBM50212640'
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212640(CHEMBL423309)
Affinity DataIC50:  37.5nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212640(CHEMBL423309)
Affinity DataIC50:  115nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212640(CHEMBL423309)
Affinity DataIC50:  230nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Enterobacter cloacae)TBA
LigandPNGBDBM50212640(CHEMBL423309)
Affinity DataIC50:  461nMAssay Description:Inhibitory activity against Enterobacter cloacae HC8 Class-I beta-lactamase enzyme type P99More data for this Ligand-Target Pair
In DepthDetails
TargetBeta-lactamase(Staphylococcus aureus)TBA
LigandPNGBDBM50212640(CHEMBL423309)
Affinity DataIC50:  461nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
In DepthDetails