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Found 2 Enz. Inhib. hit(s) with Target = 'Beta-lactamase' and Ligand = 'BDBM530966'
TargetBeta-lactamase(Pseudomonas aeruginosa)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM530966(4-[4-(2- hydroxyethyl)piperidin-1- yl]-N1-[(3R)-py...)
Affinity DataIC50:  0.130nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM530966(4-[4-(2- hydroxyethyl)piperidin-1- yl]-N1-[(3R)-py...)
Affinity DataIC50:  2.07nMAssay Description:The Class B enzyme activities were measured in the presence of the test inhibitor in a fluorescence assay against a commercially available substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent