Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with Target = 'Bifunctional protein GlmU' and Ligand = 'BDBM50365062'
TargetBifunctional protein GlmU(Escherichia coli)
Astrazeneca

LigandPNGBDBM50365062(CHEMBL1951072 | Sulfonamide, 1)
Affinity DataIC50:  2.10E+3nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
TargetBifunctional protein GlmU(Haemophilus influenzae)
Astrazeneca

LigandPNGBDBM50365062(CHEMBL1951072 | Sulfonamide, 1)
Affinity DataIC50:  7.80E+3nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Staphylococcus aureus)
Astrazeneca

LigandPNGBDBM50365062(CHEMBL1951072 | Sulfonamide, 1)
Affinity DataIC50: >2.00E+5nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Streptococcus pneumoniae)
Astrazeneca R&D Boston

Curated by ChEMBL
LigandPNGBDBM50365062(CHEMBL1951072 | Sulfonamide, 1)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Streptococcus pneumoniae acetyltransferase activity of GlmU using acetyl-CoA and glucosamine-1-phosphate after 30 mins by Ellman's meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Streptococcus pneumoniae)
Astrazeneca

LigandPNGBDBM50365062(CHEMBL1951072 | Sulfonamide, 1)
Affinity DataIC50: >2.00E+5nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed