Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Bombesin receptor subtype-3' and Ligand = 'BDBM50381918'
TargetBombesin receptor subtype-3(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50381918(CHEMBL2023113)
Affinity DataIC50: 0.5nMAssay Description:Displacement of 125I-dY-peptide from human BRS3 expressed in NFAT-CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50381918(CHEMBL2023113)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human BRS3 expressed in human HEK293AEQ cells measured for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50381918(CHEMBL2023113)
Affinity DataEC50:  22nMAssay Description:Agonist activity at mouse BRS3 expressed in human HEK293AEQ cells measured for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed