Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Bombesin receptor subtype-3' and Ligand = 'BDBM50400252'
TargetBombesin receptor subtype-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400252(CHEMBL2179913)
Affinity DataIC50: 5.80nMAssay Description:Displacement of [125I]-[D-Tyr6,beta-Ala11,Phe13,Nle14]-Bombesin(6-14) from human BRS3 expressed in CHO cells expressing NFAT after 2 hrs by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50400252(CHEMBL2179913)
Affinity DataEC50:  199nMAssay Description:Agonist activity at human BRS3 expressed in HEK293 cells expressing aequorin measured for 30 secs by bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50400252(CHEMBL2179913)
Affinity DataEC50:  377nMAssay Description:Agonist activity at mouse BRS3 expressed in HEK293 cells expressing aequorin measured for 30 secs by bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed