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Found 3 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 3' and Ligand = 'BDBM439497'
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Abbvie

Curated by ChEMBL
LigandPNGBDBM439497(US10633379, Example 35 | US10633379, Example 82)
Affinity DataKi:  4.90nMAssay Description:Inhibition of BRD3 BD2 (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Abbvie

Curated by ChEMBL
LigandPNGBDBM439497(US10633379, Example 35 | US10633379, Example 82)
Affinity DataKi:  3.14E+3nMAssay Description:Inhibition of BRD3 BD1 (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Abbvie

Curated by ChEMBL
LigandPNGBDBM439497(US10633379, Example 35 | US10633379, Example 82)
Affinity DataIC50:  0.880nMAssay Description:Inhibition of C-terminal His6-tagged BRD3 BD2 (unknown origin) using H-YSGRGK(Ac)GGK(Ac)GLGK(Ac)-GGAK(Ac)RHRK-Biotin-OH as substrate incubated for 1 ...More data for this Ligand-Target Pair
In DepthDetails PubMed