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Found 5 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM50593635'
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50593635(CHEMBL5205867)
Affinity DataKd:  2nMAssay Description:Binding affinity to BRD4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50593635(CHEMBL5205867)
Affinity DataKd:  301nMAssay Description:pA2 for NK2 receptor of rabbit pulmonary arteryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50593635(CHEMBL5205867)
Affinity DataKd:  2nMAssay Description:Binding affinity to BDR4- BD2 (unknown origin) assessed as dissociation constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50593635(CHEMBL5205867)
Affinity DataKd:  301nMAssay Description:Binding affinity to BDR4-BD1 (unknown origin) assessed as dissociation constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50593635(CHEMBL5205867)
Affinity DataKd:  2nMAssay Description:pA2 for NK2 receptor of rabbit pulmonary arteryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed