Found 8 Enz. Inhib. hit(s) with Target = 'C-C chemokine receptor type 1' and Ligand = 'BDBM50436256'
Affinity DataIC50: 0.800nMAssay Description:Binding affinity to human CCR1More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of RANTES-induced chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MIP1alpha-induced chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of MPIF-1-induced chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of HCC-1-induced chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:Antagonist activity at human CCR1 assessed as inhibition of ieukotactin-1-induced chemotaxisMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Antagonist activity at CCR1 in whole blood (unknown origin) assessed as inhibition of MIP1alpha-induced upregulation of beta2-integrin CD11bMore data for this Ligand-Target Pair
Affinity DataIC50: 54nMAssay Description:Antagonist activity at CCR1 in whole blood (unknown origin) assessed as inhibition of LKN1-induced upregulation of beta2-integrin CD11bMore data for this Ligand-Target Pair