Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'C-C chemokine receptor type 2' and Ligand = 'BDBM50268369'
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50268369(CHEMBL451340 | N-(2-((1S,2R,4R)-4-(benzylamino)-2-...)
Affinity DataIC50:  8.40nMAssay Description:Displacement of [125I]MCP1 from CCR2 in human PBMC by millipore filter plate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50268369(CHEMBL451340 | N-(2-((1S,2R,4R)-4-(benzylamino)-2-...)
Affinity DataIC50:  12.7nMAssay Description:Antagonist activity at CCR2 in human PBMC assessed as MCP1-induced chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed