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Found 5 Enz. Inhib. hit(s) with Target = 'C-X-C chemokine receptor type 4' and Ligand = 'BDBM50246956'
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50246956(1,3-dicyclohexyl-2-((5,6-dihydroimidazo[2,1-b]thia...)
Affinity DataIC50:  11nMAssay Description:Activity at CXCR4 in human CEM cells assessed as inhibition of CXCL12-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Rattus norvegicus (Rat))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50246956(1,3-dicyclohexyl-2-((5,6-dihydroimidazo[2,1-b]thia...)
Affinity DataIC50:  29nMAssay Description:Activity at CXCR4 in rat IR983F cells assessed as inhibition of CXCL12-induced cell migrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50246956(1,3-dicyclohexyl-2-((5,6-dihydroimidazo[2,1-b]thia...)
Affinity DataIC50:  48nMAssay Description:Displacement of [125I]CXCL12 from CXCR4 in human CEM cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Rattus norvegicus (Rat))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50246956(1,3-dicyclohexyl-2-((5,6-dihydroimidazo[2,1-b]thia...)
Affinity DataIC50:  55nMAssay Description:Displacement of [125I]CXCL12 from CXCR4 in rat IR983F cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50246956(1,3-dicyclohexyl-2-((5,6-dihydroimidazo[2,1-b]thia...)
Affinity DataIC50:  58nMAssay Description:Activity at CXCR4 in human Jurkat T cells assessed as inhibition of CXCL12-induced cell migrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed