Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'C-X-C chemokine receptor type 4' and Ligand = 'BDBM50333884'
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50333884((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-N-(4-(ami...)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at CXCR4 in human CEM-CCRF cells expressing CD4 assessed as inhibition of SDF-1-induced Ca2+ signalingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50333884((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-N-(4-(ami...)
Affinity DataIC50:  88.9nMAssay Description:Displacement of [125I]SDF-1 from CXCR4 in human CEM-CCRF cells expressing CD4 by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed