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Found 2 Enz. Inhib. hit(s) with Target = 'C-X-C chemokine receptor type 6' and Ligand = 'BDBM50539439'
TargetC-X-C chemokine receptor type 6(Homo sapiens)
Sanford Burnham Prebys Medical Discovery Institute

Curated by ChEMBL
LigandPNGBDBM50539439(CHEMBL4646463)
Affinity DataIC50:  2.10E+3nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of CXCL16-induced beta-arrestin recruitment by DiscoveRx cell based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 6(Homo sapiens)
Sanford Burnham Prebys Medical Discovery Institute

Curated by ChEMBL
LigandPNGBDBM50539439(CHEMBL4646463)
Affinity DataIC50:  1.47E+4nMAssay Description:Antagonist activity at Prolink-tagged human CXCR6 receptor assessed as inhibition of forskolin-induced cAMP accumulation by DiscoveRx cell based assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed