Found 4 Enz. Inhib. hit(s) with Target = 'C3a anaphylatoxin chemotactic receptor' and Ligand = 'BDBM50388995' TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 26.3nMAssay Description:Antagonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant compound preincubat...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataIC50: 1.12E+3nMAssay Description:Antagonist activity at C3a receptor in dbcAMP differentiated human U937 cells assessed as inhibition of increase in intracellular calcium compound pr...More data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 35.5nMAssay Description:Agonist activity at human C3a receptor expressed in RBL-2H3 cells assessed as beta-hexosaminidase activity in cell supernatant by degranulation assayMore data for this Ligand-Target Pair
TargetC3a anaphylatoxin chemotactic receptor(Homo sapiens (Human))
Princeton University
Curated by ChEMBL
Princeton University
Curated by ChEMBL
Affinity DataEC50: 661nMAssay Description:Partial agonist activity at C3a receptor in dbcAMP differentiated human U937 cells assessed as increase in intracellular calcium using Fluo-R stainin...More data for this Ligand-Target Pair
