Found 1 Enz. Inhib. hit(s) with Target = 'Calcium release-activated calcium channel protein/Stromal interaction molecule 1' and Ligand = 'BDBM50575331'
TargetCalcium release-activated calcium channel protein/Stromal interaction molecule 1(Homo sapiens (Human))
Lupin
Curated by ChEMBL
Lupin
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Inhibition of Orai1/STIM1 (unknown origin) expressed in HEK293 cells assessed as reduction in Ca2+-release activated Ca2+ entry current by manual pat...More data for this Ligand-Target Pair