Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Calpain-2 catalytic subunit' and Ligand = 'BDBM50039994'
TargetCalpain-2 catalytic subunit(Homo sapiens (Human))
Alkermes

Curated by ChEMBL
LigandPNGBDBM50039994(CHEMBL419898 | [(S)-1-(1-Ethylcarbamoyl-butylcarba...)
Affinity DataKi:  42nMAssay Description:Tested for inhibitory activity on porcine calpain 2 from kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Bos taurus)
Alkermes

Curated by ChEMBL
LigandPNGBDBM50039994(CHEMBL419898 | [(S)-1-(1-Ethylcarbamoyl-butylcarba...)
Affinity DataKi:  50nMAssay Description:Tested for inhibitory activity on bovine calpain 2 from heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-2 catalytic subunit(Homo sapiens (Human))
Alkermes

Curated by ChEMBL
LigandPNGBDBM50039994(CHEMBL419898 | [(S)-1-(1-Ethylcarbamoyl-butylcarba...)
Affinity DataKi:  73nMAssay Description:Tested for inhibitory activity on human calpain 2 from placentaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed