Affinity DataKi: 100nMAssay Description:Displacement of [3H]-CP-55,940 from rat forebrain membrane which expresses Cannabinoid receptor 1 in the presence of PMSFMore data for this Ligand-Target Pair
Affinity DataKi: 470nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 472nMAssay Description:Binding affinity to rat CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 472nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in Wistar rat brain incubated for 60 mins by radioactive filter binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 472nMAssay Description:Binding affinity to CB1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 480nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK-293-EBNA cell membranes after 90 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity to CB1R (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Potency at CB1 receptor in rat brain by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 23nMAssay Description:Agonist activity at CB1 receptor expressed in NG108-15 cells assessed as increase in intracellular free calcium concentrationsMore data for this Ligand-Target Pair