Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50170333'
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170333(JWH-302 | 2-(3-methoxyphenyl)-1-(1-pentyl-1H-indol...)
Affinity DataEC50:  29.3nMAssay Description:Effective concentration for stimulation of [35S]GTP-gamma-S binding at CB1 receptor in presence of 10 uM WIN-55212-2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170333(JWH-302 | 2-(3-methoxyphenyl)-1-(1-pentyl-1H-indol...)
Affinity DataKi:  17nMAssay Description:Binding affinity to displace [3H]CP-55940 from CB1 receptor of rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50170333(JWH-302 | 2-(3-methoxyphenyl)-1-(1-pentyl-1H-indol...)
Affinity DataKi:  17.0nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed