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Found 3 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50316513'
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50316513(CHEMBL1096182 | N-((4R)-6-(4-chlorophenyl)-7-(2,4-...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of rat cannabinoid CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50316513(CHEMBL1096182 | N-((4R)-6-(4-chlorophenyl)-7-(2,4-...)
Affinity DataIC50:  1nMAssay Description:Displacement of [3H]CP55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50316513(CHEMBL1096182 | N-((4R)-6-(4-chlorophenyl)-7-(2,4-...)
Affinity DataEC50:  5.80nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB1 receptor expressed in CHO cellssassessed as inhibition of forskolin-stimulated increase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed