Affinity DataIC50: 0.700nMAssay Description:Inhibition of rat cannabinoid CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]CP55940 from human recombinant cannabinoid CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 5.80nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB1 receptor expressed in CHO cellssassessed as inhibition of forskolin-stimulated increase...More data for this Ligand-Target Pair