Affinity DataKi: 37nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 99.3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >2.50E+4nMAssay Description:Antagonist activity at human brain CB1 receptor assessed as inhibition for [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity at rat brain CB1 receptor assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair