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Found 4 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50380886'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380886(CHEMBL2019082)
Affinity DataKi:  3.06E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor membrane fractionsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380886(CHEMBL2019082)
Affinity DataKi:  3.06E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380886(CHEMBL2019082)
Affinity DataIC50: >2.00E+3nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cells assessed as increase in forskolin-induced cAMP levels after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50380886(CHEMBL2019082)
Affinity DataIC50: >2.00E+3nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP release after 25 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed