Affinity DataIC50: 40nMAssay Description:Allosteric antagonist activity at mouse CB1 receptor by GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Allosteric antagonist activity at mouse CB1 receptor by GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataIC50: 169nMAssay Description:Allosteric antagonist activity at human CB1 receptor by Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataIC50: 169nMAssay Description:Allosteric antagonist activity at human CB1 receptor by Ca2+ assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.40nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.40nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorMore data for this Ligand-Target Pair