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Found 3 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50006261'
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50006261(CHEMBL3234698)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]-CP55940 from rat CB2 receptor expressed in CHO-K1 cells by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50006261(CHEMBL3234698)
Affinity DataKi:  27nMAssay Description:Agonist activity at human CB2 receptor assessed as inhibition of forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50006261(CHEMBL3234698)
Affinity DataEC50:  0.470nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed