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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50116909'
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50116909(CHEMBL3613101)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor transfected in HEK293EBNA cell membranes after 90 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50116909(CHEMBL3613101)
Affinity DataIC50:  1.82E+3nMAssay Description:Antagonist/inverse agonist activity at human CB2 receptor transfected in Chem4 cell membranes after 30 mins by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed