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Found 4 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50382752'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50382752(CHEMBL2023580)
Affinity DataKi:  885nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50382752(CHEMBL2023580)
Affinity DataKi:  885nMAssay Description:Binding affinity to CB2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50382752(CHEMBL2023580)
Affinity DataKi:  885nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor membrane fractionsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50382752(CHEMBL2023580)
Affinity DataIC50:  800nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells assessed as increase in forskolin-induced cAMP levels after 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed