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Found 3 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50399121'
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399121(CHEMBL2179751)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399121(CHEMBL2179751)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cells incubated for 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50399121(CHEMBL2179751)
Affinity DataEC50:  28.3nMAssay Description:Inverse agonist activity at human CB2 receptor expressed in CHO cells assessed as increase in forskolin-induced cAMP accumulation incubated for 45 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed