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Found 1 Enz. Inhib. hit(s) with Target = 'Carboxylic ester hydrolase' and Ligand = 'BDBM10525'
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Universita Degli Studi Di Siena

LigandPNGBDBM10525(N-[6-(1,2,3,4-tetrahydroacridin-9-ylsulfanyl)hexyl...)
Affinity DataKi:  30nM ΔG°:  -42.9kJ/molepH: 8.0 T: 2°CAssay Description:Inhibition of enzyme activity was measured over a substrate concentration range of 0.01-30 mM and at least six inhibitor concentrations to determine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed