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Found 3 Enz. Inhib. hit(s) with Target = 'Cholecystokinin receptor type A' and Ligand = 'BDBM50056102'
TargetCholecystokinin receptor type A(Homo sapiens (Human))
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50056102((R)-1-(1-(3,3-dimethyl-2-oxobutyl)-2-oxo-5-(pyridi...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]L-364718 from human recombinant CCK1 receptor expressed in CHOK1 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
James Black Foundation

Curated by ChEMBL
LigandPNGBDBM50056102((R)-1-(1-(3,3-dimethyl-2-oxobutyl)-2-oxo-5-(pyridi...)
Affinity DataKi:  398nMAssay Description:Displacement of [125I]BH-CCK-8S from CC1 receptor expressed in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50056102((R)-1-(1-(3,3-dimethyl-2-oxobutyl)-2-oxo-5-(pyridi...)
Affinity DataIC50:  502nMAssay Description:Inhibitory concentration against radioligand [3 H]L-364,718 binding to gastrin/Cholecystokinin type A receptor from rat pancreasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed