Found 3 Enz. Inhib. hit(s) with Target = 'Cholecystokinin receptor type A' and Ligand = 'BDBM50060322'
Affinity DataKi: 0.620nMAssay Description:Inhibition of [3H]-pCCK-8 specific binding to Cholecystokinin type A receptor of rat pancreasMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)
Curated by ChEMBL
Instituto De QuíMica MéDica (Csic)
Curated by ChEMBL
Affinity DataIC50: 6.85E+3nMAssay Description:Inhibition of CCK binding to Cos-7 cells expressing human cholecystokinin 1 receptorMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Instituto De QuíMica MéDica (Csic)
Curated by ChEMBL
Instituto De QuíMica MéDica (Csic)
Curated by ChEMBL
Affinity DataIC50: 2.09E+4nMAssay Description:Inhibition of CCK-Induced inositol phosphate production in Cos-7 cells expressing human CCK1RMore data for this Ligand-Target Pair