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Found 4 Enz. Inhib. hit(s) with Target = 'Cholecystokinin receptor type A' and Ligand = 'BDBM50329181'
TargetCholecystokinin receptor type A(RAT)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50329181(3-(6-(2-(benzyl(isopropyl)amino)-2-oxoethyl)-5-oxo...)
Affinity DataIC50:  17nMAssay Description:Displacement of [125I]CCK8 from rat CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50329181(3-(6-(2-(benzyl(isopropyl)amino)-2-oxoethyl)-5-oxo...)
Affinity DataIC50:  49.3nMAssay Description:Displacement of [125I]CCK8 from human CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50329181(3-(6-(2-(benzyl(isopropyl)amino)-2-oxoethyl)-5-oxo...)
Affinity DataEC50:  428nMAssay Description:Agonist activity at rat CCK1 receptor expressed in CHO cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50329181(3-(6-(2-(benzyl(isopropyl)amino)-2-oxoethyl)-5-oxo...)
Affinity DataEC50:  645nMAssay Description:Agonist activity at human CCK1 receptor expressed in CHO cells assessed as induction of calcium release by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed