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Found 6 Enz. Inhib. hit(s) with Target = 'Cholesteryl ester transfer protein' and Ligand = 'BDBM50094514'
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Universidade Federal Da Bahia

Curated by ChEMBL
LigandPNGBDBM50094514(1,1,1-Trifluoro-3-[(3-phenoxy-phenyl)-(3-trifluoro...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Universidade Federal Da Bahia

Curated by ChEMBL
LigandPNGBDBM50094514(1,1,1-Trifluoro-3-[(3-phenoxy-phenyl)-(3-trifluoro...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of recombinant human CETP-mediated transfer of [3H]-CE from HDL to LDLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Oryctolagus cuniculus)
Al-Zaytoonah Private University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50094514(1,1,1-Trifluoro-3-[(3-phenoxy-phenyl)-(3-trifluoro...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of CETP in rabbit serum after 1 hr by fluorescent cholesteryl esters transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Universidade Federal Da Bahia

Curated by ChEMBL
LigandPNGBDBM50094514(1,1,1-Trifluoro-3-[(3-phenoxy-phenyl)-(3-trifluoro...)
Affinity DataIC50:  1.00E+3nMAssay Description:Concentration required for 50% inhibition of cholesteryl ester transfer protein in presence of buffer.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Universidade Federal Da Bahia

Curated by ChEMBL
LigandPNGBDBM50094514(1,1,1-Trifluoro-3-[(3-phenoxy-phenyl)-(3-trifluoro...)
Affinity DataIC50:  4.00E+4nMAssay Description:Tested for inhibiting CETP-mediated transfer of [3H]-CE from HDL to LDL in vitro under buffered assay conditions in human serum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Universidade Federal Da Bahia

Curated by ChEMBL
LigandPNGBDBM50094514(1,1,1-Trifluoro-3-[(3-phenoxy-phenyl)-(3-trifluoro...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of cholesteryl ester transfer protein in presence of human serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed