Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with Target = 'Cholesteryl ester transfer protein' and Ligand = 'BDBM50100997'
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Universidade Federal Da Bahia

Curated by ChEMBL
LigandPNGBDBM50100997(1,1,1-Trifluoro-3-[(3-furan-2-yl-benzyl)-(3-phenox...)
Affinity DataIC50:  480nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Universidade Federal Da Bahia

Curated by ChEMBL
LigandPNGBDBM50100997(1,1,1-Trifluoro-3-[(3-furan-2-yl-benzyl)-(3-phenox...)
Affinity DataIC50:  480nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]-cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Oryctolagus cuniculus)
Al-Zaytoonah Private University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50100997(1,1,1-Trifluoro-3-[(3-furan-2-yl-benzyl)-(3-phenox...)
Affinity DataIC50:  480nMAssay Description:Inhibition of CETP in rabbit serum after 1 hr by fluorescent cholesteryl esters transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Universidade Federal Da Bahia

Curated by ChEMBL
LigandPNGBDBM50100997(1,1,1-Trifluoro-3-[(3-furan-2-yl-benzyl)-(3-phenox...)
Affinity DataIC50:  480nMAssay Description:Inhibition of recombinant human CETP in buffer assessed as transfer of [3H]-cholesteryl ester from HDL donor particles to LDL acceptor particlesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Universidade Federal Da Bahia

Curated by ChEMBL
LigandPNGBDBM50100997(1,1,1-Trifluoro-3-[(3-furan-2-yl-benzyl)-(3-phenox...)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of recombinant human CETP mediated transfer of [3H]-cholesteryl ester from HDL to LDLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed