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Found 4 Enz. Inhib. hit(s) with Target = 'Cholesteryl ester transfer protein' and Ligand = 'BDBM50101002'
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101002(1,1,1-Trifluoro-3-[(4-fluoro-3-furan-2-yl-benzyl)-...)
Affinity DataIC50:  720nMAssay Description:In vitro human CETP inhibitory activity assessed by measuring the rate of [3H]-cholesteryl ester ([3H]-CE) from HDL donor particles to LDL acceptor p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Oryctolagus cuniculus)
Al-Zaytoonah Private University Of Jordan

Curated by ChEMBL
LigandPNGBDBM50101002(1,1,1-Trifluoro-3-[(4-fluoro-3-furan-2-yl-benzyl)-...)
Affinity DataIC50:  720nMAssay Description:Inhibition of CETP in rabbit serum after 1 hr by fluorescent cholesteryl esters transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101002(1,1,1-Trifluoro-3-[(4-fluoro-3-furan-2-yl-benzyl)-...)
Affinity DataIC50:  720nMAssay Description:Inhibition of CETPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50101002(1,1,1-Trifluoro-3-[(4-fluoro-3-furan-2-yl-benzyl)-...)
Affinity DataIC50:  4.90E+4nMAssay Description:In vitro human CETP inhibitory activity assessed by measuring the rate of [3H]-cholesteryl ester ([3H]-CE) from HDL donor particles to LDL acceptor p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed