Found 4 Enz. Inhib. hit(s) with Target = 'Cholesteryl ester transfer protein' and Ligand = 'BDBM50101002'
Affinity DataIC50: 720nMAssay Description:In vitro human CETP inhibitory activity assessed by measuring the rate of [3H]-cholesteryl ester ([3H]-CE) from HDL donor particles to LDL acceptor p...More data for this Ligand-Target Pair
TargetCholesteryl ester transfer protein(Oryctolagus cuniculus)
Al-Zaytoonah Private University Of Jordan
Curated by ChEMBL
Al-Zaytoonah Private University Of Jordan
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of CETP in rabbit serum after 1 hr by fluorescent cholesteryl esters transfer assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+4nMAssay Description:In vitro human CETP inhibitory activity assessed by measuring the rate of [3H]-cholesteryl ester ([3H]-CE) from HDL donor particles to LDL acceptor p...More data for this Ligand-Target Pair