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Found 4 Enz. Inhib. hit(s) with Target = 'Cholinesterase' and Ligand = 'BDBM50246979'
TargetCholinesterase(Homo sapiens (Human))
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50246979(CHEMBL4105611 | US20230331674, Table 1.1)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of recombinant human BChE using butyrylthiocholine iodide as substrate preincubated for 300 secs followed by substrate addition measured f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCholinesterase(Homo sapiens (Human))
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50246979(CHEMBL4105611 | US20230331674, Table 1.1)
Affinity DataIC50:  4.90nMAssay Description:The inhibitory potencies against huBChE and murine AChE (mAChE) were determined for all of these synthesized compounds using the method of Ellman (El...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCholinesterase(Homo sapiens (Human))
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50246979(CHEMBL4105611 | US20230331674, Table 1.1)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of recombinant human BChE using butyrylthiocholine as substrate measured after 300 secs by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCholinesterase(Homo sapiens (Human))
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50246979(CHEMBL4105611 | US20230331674, Table 1.1)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of human recombinant BChE pre-incubated for 300 secs before substrate addition by Ellman's methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB