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Found 3 Enz. Inhib. hit(s) with Target = 'Citron Rho-interacting kinase' and Ligand = 'BDBM24773'
TargetCitron Rho-interacting kinase(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM24773(AMG 706 | AMG-706 | Motesanib | N-(3,3-dimethyl-1,...)
Affinity DataKd:  300nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetCitron Rho-interacting kinase(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM24773(AMG 706 | AMG-706 | Motesanib | N-(3,3-dimethyl-1,...)
Affinity DataKd:  300nMAssay Description:Binding constant for CIT kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCitron Rho-interacting kinase(Homo sapiens (Human))
Ambit Biosciences

Curated by PubChem BioAssay
LigandPNGBDBM24773(AMG 706 | AMG-706 | Motesanib | N-(3,3-dimethyl-1,...)
Affinity DataKd:  300nMAssay Description:Binding constant for CIT kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed