Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Cyclin-A2/Cyclin-dependent kinase 2' and Ligand = 'BDBM572061'
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572061((R)-N-(4-(3-(quinazolin-2- ylamino)pyrrolidine-1- ...)
Affinity DataIC50:  550nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Kinnate Biopharma

US Patent
LigandPNGBDBM572061((R)-N-(4-(3-(quinazolin-2- ylamino)pyrrolidine-1- ...)
Affinity DataIC50:  5.50E+3nMAssay Description:A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the protein kinase. All kinase assays ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent