Affinity DataIC50: 7nMAssay Description:Inhibition of GST-tagged human CDK12/Cyclin K expressed in Sf9 cells using RBER-IRStide peptide as substrate in presence of ATP and [gamma33-P] ATP b...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human CDK12 (696 to 1082 residues)/human cyclinK (1 to 267 residues) using pol2 CTD-peptide substrate and [gammaP]ATP by scintillation ...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of CDK12 (unknown origin)More data for this Ligand-Target Pair