Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 12' and Ligand = 'BDBM50588263'
TargetCyclin-dependent kinase 12(Homo sapiens)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50588263(CHEMBL5198038)
Affinity DataIC50:  40nMAssay Description:Inhibition of CDK12 (unknown origin) using FITC-X-GSRTPMY-NH2 as substrate preincubated for 10 mins followed by substrate addition and measured after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCyclin-dependent kinase 12(Homo sapiens)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50588263(CHEMBL5198038)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of CDK12 (unknown origin) using FITC-X-GSRTPMY-NH2 as substrate preincubated for 10 mins followed by substrate addition and measured after...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed