Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 2/G1/S-specific cyclin-E1' and Ligand = 'BDBM370256'
LigandChemical structure of BindingDB Monomer ID 370256BDBM370256(US10233188, Example 143 | BDBM467151)
Affinity DataKi:  2.42nMAssay Description:The purpose of the CDK2/Cyclin E1 assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a flu...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/27/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 370256BDBM370256(US10233188, Example 143 | BDBM467151)
Affinity DataKi:  2.42nMAssay Description:The purpose of the CDK2/Cyclin E1 assay is to evaluate the inhibition (% inhibition, Kiapp and Ki values) of small molecule inhibitors by using a flu...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
6/1/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 370256BDBM370256(US10233188, Example 143 | BDBM467151)
Affinity DataKi:  2.42nMAssay Description:The mobility shift assay electrophoretically separates the fluorescently labeled peptides (substrate and phosphorylated product) following the kinase...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
10/17/2022
Entry Details
US Patent